28 Apr 2008

Biochemical Pharmacology :Vol 75, Issue 8

Commentary

2.
Anti-inflammatory interventions of NF-κB signaling: Potential applications and risks Pages 1567-1579 Senftleben Uwe

Antibiotics and Chemotherapeutics

3.
Accumulation of the antimalarial microtubule inhibitors trifluralin and vinblastine by Plasmodium falciparum Pages 1580-1587 Julie Ann Naughton, Ruth Hughes, Patrick Bray and Angus Bell


4.
Structure–activity relationship for adenosine kinase from Mycobacterium tuberculosis: II. Modifications to the ribofuranosyl moiety Pages 1588-1600 Mary C. Long, Sue C. Shaddix, Omar Moukha-Chafiq, Joseph A. Maddry, Lisa Nagy and William B. Parker


5.
Thiopurine analogues inhibit papain-like protease of severe acute respiratory syndrome coronavirus Pages 1601-1609 Chi-Yuan Chou, Chia-Hui Chien, Yu-San Han, Mojca Trstenjak Prebanda, Hsing-Pang Hsieh, Boris Turk, Gu-Gang Chang and Xin Chen


6.
Effect of AZT on thymidine phosphorylation in cultured H9c2, U-937, and Raji cell lines Pages 1610-1615 Matthew D. Lynx, Bae-Kwang Kang and Edward E. McKee


7.
Modulatory effects of 5-fluorouracil on the rhythmic expression of circadian clock genes: A possible mechanism of chemotherapy-induced circadian rhythm disturbances Pages 1616-1622 Hideyuki Terazono, Ahmed Hamdan, Naoya Matsunaga, Naoto Hayasaka, Hiroaki Kaji, Takashi Egawa, Kazutaka Makino, Yasufumi Shigeyoshi, Satoru Koyanagi and Shigehiro Ohdo

Cardiovascular Pharmacology

8.
Transactivation of epidermal growth factor receptor in vascular and renal systems in rats with experimental hyperleptinemia: Role in leptin-induced hypertension Pages 1623-1638 Anna Jamroz-Wiśniewska, Grażyna Wójcicka, Ewelina Łowicka, Marta Książek and Jerzy Bełtowski


9.
Domain mapping of a claudin-4 modulator, the C-terminal region of C-terminal fragment of Clostridium perfringens enterotoxin, by site-directed mutagenesis Pages 1639-1648 Azusa Takahashi, Eriko Komiya, Hideki Kakutani, Takeshi Yoshida, Makiko Fujii, Yasuhiko Horiguchi, Hiroyuki Mizuguchi, Yasuo Tsutsumi, Shin-ichi Tsunoda, Naoya Koizumi, Katsuhiro Isoda, Kiyohito Yagi, Yoshiteru Watanabe and Masuo Kondoh


10.
Insulin therapy restores impaired function and expression of P-glycoprotein in blood–brain barrier of experimental diabetes Pages 1649-1658 Haiyan Liu, Xiaodong Liu, Lee Jia, Yuchun Liu, Huiwen Yang, Guangji Wang and Lin Xie

Pharmacokinetics and Drug Metabolism

11.
Role of proline 1150 in functional interactions between the membrane spanning domains and nucleotide binding domains of the MRP1 (ABCC1) transporter Pages 1659-1669 Isabelle J. Létourneau, Akio Nakajima, Roger G. Deeley and Susan P.C. Cole


12.
Quercetin pretreatment increases the bioavailability of pioglitazone in rats: Involvement of CYP3A inhibition Pages 1670-1676 Sudhir N. Umathe, Pankaj V. Dixit, Vijendra kumar, Kuldeep U. Bansod and Manish M. Wanjari


13.
Changes in maternal liver Cyp2c and Cyp2d expression and activity during rat pregnancy Pages 1677-1687 Leslie J. Dickmann, Suzanne Tay, Tauri D. Senn, Huixia Zhang, Anthony Visone, Jashvant D. Unadkat, Mary F. Hebert and Nina Isoherranen

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